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USE OF CATECHOLAMINES AND RELATED COMPOUNDS AS ANT

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专利名称:USE OF CATECHOLAMINES AND RELATED

COMPOUNDS AS ANTI-ANGIOGENICAGENTS

发明人:KONISHI, Yasuo,MAGOON,

Joanne,JARUSSOPHON, Suwatchai

申请号:EP08706338.4申请日:20080129公开号:EP2117524B8公开日:20190925

摘要:A catecholamine or related compound having (S)-configuration at -carbon, aphysiologically tolerated salt thereof, a prodrug thereof, a physiologically functionalderivative thereof or any mixture thereof and having a lipophilicity greater than (S)-noradrenaline has use as an anti-angiogenic agent. A catecholamine or related compoundin which a -hydroxy group has been modified are also anti-angiogenic. The anti-angiogenicagent is preferably a compound of formula (I) or (II) a physiologically tolerated saltthereof, a prodrug thereof, a physiologically functional derivative thereof or any mixturethereof.

申请人:National Research Council of Canada

代理机构:Glück Kritzenberger Patentanwälte PartGmbB

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